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Haggarty SJ, Koeller KM, Wong JC, Butcher RA, Schreiber SL. Multidimensional chemical genetic analysis of diversity-oriented synthesis-derived deacetylase inhibitors using cell-based assays. Chem Biol. 2003;10(5):383-96.
Koeller KM, Haggarty SJ, Perkins BD, et al. Chemical genetic modifier screens: small molecule trichostatin suppressors as probes of intracellular histone and tubulin acetylation. Chem Biol. 2003;10(5):397-410.
Koehler AN, Shamji AF, Schreiber SL. Discovery of an inhibitor of a transcription factor using small molecule microarrays and diversity-oriented synthesis. J Am Chem Soc. 2003;125(28):8420-1. doi:10.1021/ja0352698
Burke MD, Berger EM, Schreiber SL. Generating diverse skeletons of small molecules combinatorially. Science. 2003;302(5645):613-8. doi:10.1126/science.1089946
Wong JC, Sternson SM, Louca JB, Hong R, Schreiber SL. Modular synthesis and preliminary biological evaluation of stereochemically diverse 1,3-dioxanes. Chem Biol. 2004;11(9):1279-91. doi:10.1016/j.chembiol.2004.07.012
Burke MD, Berger EM, Schreiber SL. A synthesis strategy yielding skeletally diverse small molecules combinatorially. J Am Chem Soc. 2004;126(43):14095-104. doi:10.1021/ja0457415
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Lo MMC, Neumann CS, Nagayama S, Perlstein EO, Schreiber SL. A library of spirooxindoles based on a stereoselective three-component coupling reaction. J Am Chem Soc. 2004;126(49):16077-86. doi:10.1021/ja045089d
Kumar N, Kiuchi M, Tallarico JA, Schreiber SL. Small-molecule diversity using a skeletal transformation strategy. Org Lett. 2005;7(13):2535-8. doi:10.1021/ol0504345